Evaluation of 2,3-Dihydro-1,5-benzothiazepine Derivatives as Potential Tyrosinase Inhibitors: In Vitro and In Silico Studies

Munirah M. Al-Rooqi; Amina Sadiq; Rami J. Obaid; Zaman Ashraf; Yasir Nazir; Rabab S. Jassas; Nafeesa Naeem; Meshari A. Alsharif; Syed Wadud Ali Shah; Ziad Moussa; Ehsan Ullah Mughal; Abdel-Rahman Farghaly; Saleh A. Ahmed

doi:10.1021/acsomega.3c01566

journal article Open Access May 04, 2023

Evaluation of 2,3-Dihydro-1,5-benzothiazepine Derivatives as Potential Tyrosinase Inhibitors: In Vitro and In Silico Studies

Munirah M. Al-Rooqi Amina Sadiq

Rami J. Obaid Zaman Ashraf

Yasir Nazir

Rabab S. Jassas Nafeesa Naeem

Meshari A. Alsharif Syed Wadud Ali Shah Ziad Moussa

Ehsan Ullah Mughal

Abdel-Rahman Farghaly Saleh A. Ahmed

ACS Omega Vol. 8 No. 19 pp. 17195-17208 · American Chemical Society (ACS)

View at Publisher Save 10.1021/acsomega.3c01566

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Citations

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References

Details

Published: May 04, 2023
Vol/Issue: 8(19)
Pages: 17195-17208
License: View

Authors

M

Munirah M. Al-Rooqi

Department of Chemistry, Faculty of Applied Sciences, Umm Al-Qura University, Makkah 21955, Saudi Arabia

A

Amina Sadiq

Department of Chemistry, Govt. College Women University, Sialkot 51300, Pakistan

R

Rami J. Obaid

Department of Chemistry, Faculty of Applied Sciences, Umm Al-Qura University, Makkah 21955, Saudi Arabia

Z

Zaman Ashraf

Department of Chemistry, Allama Iqbal Open University, Islamabad 44000, Pakistan

Y

Yasir Nazir

Department of Chemistry, Allama Iqbal Open University, Islamabad 44000, Pakistan; Department of Chemistry, University of Sialkot, Sialkot 51300, Pakistan

R

Rabab S. Jassas

Department of Chemistry, Jamoum University College, Umm Al-Qura University, Makkah 21955, Saudi Arabia

N

Nafeesa Naeem

Department of Chemistry, University of Gujrat, Gujrat 50700, Pakistan

M

Meshari A. Alsharif

Department of Chemistry, Faculty of Applied Sciences, Umm Al-Qura University, Makkah 21955, Saudi Arabia

S

Syed Wadud Ali Shah

Department of Pharmacy, University of Malakand, Chakdara Dir 18000, Khyber Pakhtunkhwa, Pakistan

Z

Ziad Moussa

Department of Chemistry, College of Science, United Arab Emirates University, P.O. Box 15551, Al Ain, Abu Dhabi, United Arab Emirates

E

Ehsan Ullah Mughal

Department of Chemistry, University of Gujrat, Gujrat 50700, Pakistan

A

Abdel-Rahman Farghaly

Department of Chemistry, College of Science, Jazan University, Jazan 114, Saudi Arabia

S

Saleh A. Ahmed

Department of Chemistry, Faculty of Applied Sciences, Umm Al-Qura University, Makkah 21955, Saudi Arabia

Funding

Higher Education Commission, Pakistan Award: NRPU-15800

United Arab Emirates University Award: G00003918

Umm Al-Qura University Award: 23UQU4320545DSR001

Cite This Article

Munirah M. Al-Rooqi, Amina Sadiq, Rami J. Obaid, et al. (2023). Evaluation of 2,3-Dihydro-1,5-benzothiazepine Derivatives as Potential Tyrosinase Inhibitors: In Vitro and In Silico Studies. ACS Omega, 8(19), 17195-17208. https://doi.org/10.1021/acsomega.3c01566

Evaluation of 2,3-Dihydro-1,5-benzothiazepine Derivatives as Potential Tyrosinase Inhibitors: In Vitro and In Silico Studies

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